Pirenperone

CAS 75444-65-4C23H24FN3O2Biochemicals & Reagents

Pirenperone (CAS: 75444-65-4; Formula: C23H24FN3O2; MW: 393.45 g/mol) is a light yellow solid compound. It acts as a selective serotonin 5-HT2A receptor antagonist. Primarily utilised in research settings, Pirenperone is a valuable tool for investigating serotonergic pathways, neurotransmission, and neuronal function. Its application is key in neuroscience research, particularly in studies related to mood disorders and behavioural science.

IUPAC: 3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2-methyl-4H-pyrido-[1,2-a] pyrimidin-4-one,R-47,465

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Pirenperone (C23H24FN3O2) — chemical structure, CAS 75444-65-4; Life Science, fine chemical supplied by Tech Serve Solutions

AntagonistsBioactive Small MoleculesBiochemicals and ReagentsCell BiologyGPCR ModulatorsGPCR ProteinsModulators and AntibodiesNeuroscienceNeurotransmissionNeurotransmission (Obesity)

01 /Applications

Neuroscience Research Tool

Pirenperone is employed in laboratory research to study the role of serotonin 5-HT2A receptors in the central nervous system. It aids in understanding neurotransmission and its involvement in various neurological processes.

Pharmacological Studies

As a selective antagonist, Pirenperone is used to probe the physiological effects of blocking 5-HT2A receptor activity. This is instrumental in developing new therapeutic strategies for conditions influenced by serotonin signalling.

Cell Signaling Investigations

Researchers utilise Pirenperone to investigate downstream signalling cascades activated by or inhibited through the 5-HT2A receptor. This helps elucidate complex cellular communication pathways.

02 /Properties

Molecular weight	393.45
Empirical formula	C23H24FN3O2
Assay	>97%
Form	solid
Colour	light yellow
Solubility	0.1 M HCl: soluble11 mg/mLmethanol: soluble2.5 mg/mL45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: soluble5.0 mg/mL

03 /Safety & handling

Protective equipment	Eyeshields, Gloves, type N95 (US), type P1 (EN143) respirator filter
Water hazard class (WGK, DE)	3

Hazard information is provided for guidance. Always consult the product Safety Data Sheet (SDS), available on request, before handling.

04 /Identifiers & registry

CAS number

75444-65-4

MDL number

MFCD00069332

05 /Additional specifications

Gene Information	human ... HTR2A(3356), HTR2B(3357), HTR2C(3358)

06 /Quality & supply

Documentation

Every batch ships with a Certificate of Analysis covering assay, identity and purity; the grade is confirmed against your enquiry. Safety Data Sheets and technical data sheets are available on request.

Supply & logistics

Samples for technical evaluation; bulk MOQ by grade and packaging. In-stock material ships in 7–10 working days, worldwide, with full export documentation.

07 /Frequently asked questions

What is Pirenperone used for?

Pirenperone is primarily used as a selective serotonin 5-HT2A receptor antagonist in research settings for neuroscience, pharmacological, and cell signaling studies.

What are the CAS number and formula for Pirenperone?

The CAS number for Pirenperone is 75444-65-4 and its empirical formula is C23H24FN3O2.

What grade and purity does Tech Serve Solutions supply?

Tech Serve Solutions supplies Pirenperone with an assay of >97%. We do not represent this product as USP, BP, or EP grade.

How should Pirenperone be handled safely?

When handling Pirenperone, it is essential to use appropriate personal protective equipment, including eyeshields, gloves, and a type N95 (US) or type P1 (EN143) respirator filter due to its potential hazards.

Is Pirenperone a controlled substance?

The provided data does not indicate that Pirenperone is a controlled substance.

How is Pirenperone packed, shipped, and exported?

Pirenperone is supplied as a light yellow solid. Tech Serve Solutions, as a global supplier, can export this chemical; please contact us for specific shipping and packing inquiries.